Falimint is a drug that has an antiseptic and local anesthetic effect. Available in the form of dragees for resorption in the oral cavity. The active substance is acetylaminonitropropoxybenzene, which inhibits the proliferation of pathogenic bacteria and eliminates sore throat. Indications for use include infections of the upper respiratory tract (pharyngitis, tonsillitis, laryngitis, tonsillitis) and oral cavity (stomatitis, gingivitis). The drug is prescribed in preparation for an instrumental examination of the pharynx and teeth. Currently, the drug is not commercially available.
Pharmacodynamics and pharmacokinetics
Pharmacodynamics
The active ingredient Falimint is an aromatic nitro compound.
The effect of the drug is similar to the effect of menthol:
- there is a feeling of pleasant coolness in the mouth and throat;
- no dryness or numbness occurs;
- breathing becomes easier immediately;
- reflex cough stops;
- mucus thins;
- pain is alleviated;
- the inflammatory process decreases;
- if there was a urge to vomit during medical manipulations in the oral cavity, they are suppressed.
Pharmacokinetics
After oral administration, Falimint is quickly absorbed. The maximum concentration of unchanged drug in plasma is achieved after 30-60 minutes.
It is excreted from the body in the form of metabolites in the urine. The maximum concentration of the altered drug in the urine is observed 2 hours after taking the tablets.
Is there an analogue of the active substance (composition)?
Having figured out where Falimint disappeared, let's move on to its analogues. Previously, Falimint could be purchased in tablet form. The composition of the pills was specified in detail in the instructions for use.
Table. Composition and active ingredient of the drug
Name | Effect |
Active substance | |
Acetylaminonitropropoxybenzene | When absorbed, it cools the throat and is effective for unproductive coughs. In the complex treatment of pharyngitis, tracheitis, bronchitis, it effectively relieves inflammation. Recommended before conducting research or taking impressions of dentures. |
Additional components | |
Sucrose | Sweetener |
Gelatin and solid fat | Filler, thickener |
Talc | Emulsifier, stabilizer |
Copovidon | Reduces the effects of toxic substances |
Colloidal silicon dioxide | Emulsifier |
Magnesium stearate | Preservative |
Surprisingly, an analogue of Falimint based on the active substance cannot be found in pharmacies. This is the only product that contains acetylaminonitropropoxybenzene. Perhaps Falimint has been discontinued, which means it is necessary to look for other solutions.
Indications for use
What Falimint tablets help with:
- diseases of the respiratory system, in which a pronounced inflammatory process is observed, in particular, tablets are taken for pharyngitis , laryngitis and tonsillitis ;
- inflammatory processes in the oral cavity, for example, stomatitis or gingivitis ;
- non-productive, dry reflex cough ;
- pronounced gag reflex during medical manipulations in the mouth and pharynx.
In most cases, in the treatment of inflammatory diseases it is used as an adjuvant.
Contraindications for which the use of tablets is prohibited
What do doctors' reviews say about the drug Falimint? Doctors report that this drug, like any other drug, has its contraindications. Don’t think that “Falimint” is a candy that helps freshen and make breathing easier. The medicine is a real medicine. The following situations are contraindications to the use of the composition:
- the period of bearing a child (throughout the entire period);
- lactation (if treatment is necessary, the issue of its termination is decided);
- the presence of hypersensitivity to the components of the drug;
- childhood.
The medicine should be used with particular caution by people with diabetes mellitus and patients with various kidney pathologies
Instructions for use of Falimint (Method and dosage)
The tablets should dissolve in the mouth. Take one tablet, no more than 10 tablets per day.
The medicine can only be used for a few days. The duration of the course is individual and should be selected by the attending physician. But if during this time the disease has not gone away, there is no need to extend the course, it is better to choose another drug.
Instructions for the use of Falimint for children have not been developed, since there is not enough information regarding the effectiveness and safety of using the medicine to treat children.
Method of use
Consumer reviews of the drug "Falimint" are mostly good. The instructions recommend using 1-2 tablets at a time. This dose will be 25-50 milligrams of the active substance. This volume in the annotation is recommended for use up to five times a day. However, doctors have a different approach to treatment with the described drug.
Doctors say that you can take no more than 10 tablets per day. Otherwise, we will already be talking about an overdose. Experts usually prescribe one capsule 6-8 times a day as needed. The drug must be dissolved slowly in the mouth. After this, you should refrain from eating and drinking for one hour.
special instructions
When treating with Falimint, you should adhere to the following recommendations:
- it is necessary to stop taking the medication if signs of a skin allergic reaction appear;
- patients with diabetes should remember that the medicine contains a certain amount of sugar (1 tablet – 0.03 bread units);
- Tablets should not be taken by persons with congenital intolerance to glucose or fructose, with glucose-galactose malabsorption or sucrose-isomaltose deficiency;
- You should not take the medicine for more than a few days.
Why Falimint disappeared from pharmacies
For many years, the drug has been effectively used for throat diseases in children and adults, and has gained well-deserved popularity among doctors and patients. Falimint helped to quickly cope with the infection and make it easier to endure the symptoms of the disease due to the local analgesic effect. However, at the end of 2022, the drug disappeared from pharmacy shelves and has not yet gone on sale.
Initially, Falimint was produced by the German pharmaceutical concern Berlin-Chemie. Then a subsidiary was created in Russia, which began to produce the drug on the domestic market. After Falimint disappeared from pharmacies, there were many theories.
Some of them referred to the economic crisis and the high cost of raw materials supplied from India and China. Others suggested a pharmaceutical conspiracy to create artificial hype around the drug in order to inflate the price. One of the first popular theories pointed to the re-registration of tablets due to a change in composition or dosage form.
When contacting the administration of Berlin-Pharma CJSC, a response was received that Falimint had been discontinued from production in Russia. They refused to announce the reason, citing non-disclosure of trade secrets. Most likely, the license from Russia was revoked as a result of problems with production and violations of the drug’s manufacturing technology. This theory is confirmed by the fact that in other countries Falimint remains on sale to this day.
>>We recommend: if you are interested in effective methods of getting rid of chronic runny nose, pharyngitis, tonsillitis, bronchitis and persistent colds, then be sure to check out this page of the site after reading this article. The information is based on the author’s personal experience and has helped many people, we hope it will help you too. Now let's return to the article.<<
Analogs
Matches by level 4 ATC code:
Suprima-ENT
Ingalipt-N
Strepsils Plus
Strepsils
Ingalipt
TheraFlu LAR
Hexoral Tabs
Lisak
Efizol
Angilex
Kameton
Anzibel
Agisept
Yox
Lugol's solution with glycerin
Lugol
Laripront
Stopangin 2A
Stopangin
Septolete Neo
Analogues of Falimint:
- Agisept;
- Vocasept;
- Hexoral Lorcept;
- Gorpils;
- Gripcold;
- Koldakt Lor Pils;
- Rinza Lorsept;
- Strepsils;
- Suprima-Lor;
- Trisils.
Caution: contraindications for use!
Contraindications:
- Pregnancy, breastfeeding period. Falimint is strictly forbidden to be used during pregnancy. Why is this happening? After all, the tablets are designed to treat sore throat, cough, and oral diseases. Medicine explains the danger of using the drug during pregnancy and breastfeeding with the following fact: Falimint has not been fully studied, and there is no required experience in using the drug during the mentioned periods of a woman’s life. For this reason, doctors do not recommend treating diseases of the throat, oral cavity and cough with this particular remedy. Moreover, nowadays there are many analogues of the drug that are safe for pregnant and lactating women.
- Individual intolerance to the drug. Before use, it is necessary to study the composition of the medicine, make sure that it does not contain components to which hypersensitivity is possible.
Falimint price
The cost of tablets in Moscow pharmacies varies. This is due to a number of reasons: retail margins, distributor or intermediary prices, rental costs, and time to purchase the medicine. The pharmacy markup is regulated by the state; its threshold should be no more than 20-25%.
You are a fairly active person who cares and thinks about your respiratory system and health in general, continue to play sports, lead a healthy lifestyle and your body will delight you throughout your life
But do not forget to undergo examinations on time, maintain your immunity, this is very important, do not overcool, avoid severe physical and strong emotional overload. Try to minimize contact with sick people; if forced contact, do not forget about protective equipment (mask, washing hands and face, cleaning the respiratory tract)
It's time to think about what you are doing wrong...
You are at risk, you should think about your lifestyle and start taking care of yourself. Physical education is required, or even better, start playing sports, choose the sport that you like most and turn it into a hobby (dancing, cycling, gym, or just try to walk more). Do not forget to treat colds and flu promptly, they can lead to complications in the lungs. Be sure to work on your immunity, strengthen yourself, and be in nature and fresh air as often as possible. Do not forget to undergo scheduled annual examinations; it is much easier to treat lung diseases in the initial stages than in advanced stages. Avoid emotional and physical overload; if possible, eliminate or minimize smoking or contact with smokers.
It's time to sound the alarm!
You are completely irresponsible about your health, thereby destroying the functioning of your lungs and bronchi, have pity on them! If you want to live a long time, you need to radically change your entire attitude towards your body. First of all, get examined by specialists such as a therapist and a pulmonologist; you need to take radical measures, otherwise everything may end badly for you. Follow all the doctors’ recommendations, radically change your life, perhaps you should change your job or even your place of residence, completely eliminate smoking and alcohol from your life, and reduce contact with people who have such bad habits to a minimum, toughen up, strengthen your immunity as much as possible spend more time in the fresh air. Avoid emotional and physical overload. Completely eliminate all aggressive products from everyday use and replace them with natural, natural remedies. Do not forget to do wet cleaning and ventilation of the room at home.
Falimint is a medicine that has an antiseptic effect, reduces sensitivity and relieves sore throat. Due to its high efficiency, for many the product has become an integral part of the first aid kit.
Why Falimint was discontinued, is it possible to buy it and what can be replaced with it - these are the main questions that concern adherents of the drug.
Composition of the drug
The following
ATC codes match. Analogues are selected according to the chemical structure of the drug and are the most suitable substitutes. Same composition, indications for use, doses of active ingredients may differ.
Ingredients: acetylaminonitropropoxybenzene
Important! Falimint stabilizes local blood flow by constricting blood vessels and reducing the activity of pro-inflammatory compounds such as histamine and bradykinin. In addition to the active ingredient, the drug contains substances to give the tablets the appropriate shape and structure
In addition to the active ingredient, the drug contains substances to give the tablets the appropriate shape and structure.
Main auxiliary components:
- sucrose;
- paraffin;
- talc.
Thanks to its simple composition and pharmacokinetics, Falimint begins to act on the mucous membrane of the upper respiratory tract, minimizing cough, within 2-3 minutes. Patients note a pleasant feeling of cold spreading to the deep parts of the pharynx and larynx.
Active ingredients in the drug "Falimint": acetylaminonitropropoxybenzene.
The composition of the dragee includes the following components: glucose syrup, simethicone emulsion, liquid paraffin and magnesium stearate.
Falimint tablets
The drug is produced in the form of biconvex round-shaped tablets, coated. The tablets are packaged in blisters of 20 pieces and are produced by the famous company Berlin-Chemie AG according to strict GMP standards. The active substance acetylaminonitropropoxybenzene is an antiseptic with a refreshing and anesthetic effect that effectively copes with an irritating cough.
Pharmacodynamics and pharmacokinetics
The tablets have antitussive, analgesic, anesthetic and antiseptic effects. They help with an unproductive, irritating cough; like menthol, they create a feeling of coolness in the mouth and throat and make breathing easier. The medicine acts gently, relieves mucus without causing dryness and numbness in the mouth. The maximum concentration of the drug is achieved in the range from 30 to 60 minutes after administration. Practically insoluble in water, the active substance is excreted in the urine in the form of intermediate metabolic products during the day.
What are Falimint tablets for?
The medicine in most cases is used as an additional remedy for diseases of the respiratory tract (tonsillitis, laryngitis, pharyngitis), accompanied by inflammation and sore throat. Indications for use are also inflammatory processes in the oral cavity (stomatitis, gingivitis), reflex dry cough. Effective for suppressing the gag reflex during medical interventions in the oral cavity and pharynx.
Overdose
Cases of overdose of Falimint have not been registered.
Latin name:
Falimint
ATC code:
R02A A20
Active ingredient:
acetylamino-nitropropoxybenzene
Manufacturer:
Berlin-Chemie/Menarini (Germany, Russian Federation)
Dispensed from the pharmacy:
Without a prescription
Storage conditions:
at temperatures up to 30°C
Shelf life:
5 l.
Falimint is an antiseptic medication with an analgesic, mild local anesthetic and antitussive effect. The therapeutic effect is achieved through suppression of the sensitivity of mucous membrane receptors in the upper parts of the respiratory system (larynx and pharynx). Thanks to this, factors of increased excitability of nerve endings that provoke the activity of the cough reflex are eliminated.
The drug does not dry out tissues and does not cause a decrease in the sensitivity of the tongue, palate or their numbness.